2017 GSK Silver Award

2016 GSK Silver Award

2016 GSK Associate Fellow

2015 GSK Exceptional Science Award

2013 GSK Exceptional Science Award

2012 GSK Exceptional Science Award

1. Xinyuan Wu, Jiayi Pan, Rufeng Fan, Yiwei Zhang, Chao Wang, Guoliang Wang, Jiaxiang Liu, Mengqing Cui, Jinfeng Yue, Rui Jin, Zhiqiang Duan, Mingyue Zheng, Lianghe Mei, Lu Zhou, Minjia Tan*, Jing Ai*, Xiaojie Lu*；Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads，J. Am. Chem. Soc. 2025，DOI: 10.1021/jacs.5c01712

2. Xinyuan Wu, Shunyao Li, Ting Liang, Qing Yu, Yiwei Zhang, Jiaxiang Liu, Kaige Li, Zijian Liu, Mengqing Cui, Yongchao Zhao, Xin Han, Rui Jin, Minjia Tan, Xiao-Hua Chen, Yujun Zhao, Mingyue Zheng, Yi Sun*, Lu Zhou*, Xiaojie Lu*; Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries, Angew. Chem. Int. Ed., 2025，https://doi.org/10.1002/anie.202505581

3. Yuhan Gui, Rui Hou, Yuchen Huang, Yu Zhou, Shihao Liu, Ling Meng, Ying Li, Fong Sang Lam, Ruoyun Ding, Yan Cao, Gang Li*, Xiaojie Lu*, Xiaoyu Li*；Discovering Cell‐Targeting Ligands and Cell‐Surface Receptors by Selection of DNA‐Encoded Chemical Libraries against Cancer Cells without Predefined Targets；Angew. Chem. Int. Ed., 2025, https://doi.org/10.1002/ange.202421172

4. Xudong Wang, Liwei Xiong, Ying Zhu, Sixiu Liu, Wenfeng Zhao, Xinyuan Wu, Mengnisa Seydimemet, Linjie Li, Peiqi Ding, Xian Lin, Jiaxiang Liu, Xuan Wang, Zhiqiang Duan, Weiwei Lu, Yanrui Suo, Mengqing Cui, Jinfeng Yue, Rui Jin, Mingyue Zheng, Yechun Xu, Lianghe Mei*, Hangchen Hu*, and Xiaojie Lu*；Covalent DNA-Encoded Library Workflow Drives Discovery of SARS-CoV-2 Nonstructural Protein Inhibitors； J. Am. Chem. Soc. 2024，146, 33983-33996.

5. Yanrui Suo,‡ Xu Qian,‡ Zhaoping Xiong, Xiaohong Liu, Chao Wang, Baiyang Mu, Xinyuan Wu,Weiwei Lu, Meiying Cui, Jiaxiang Liu, Yujie Chen, Mingyue Zheng*, and Xiaojie Lu*; Enhancing the Predictive Power of Machine Learning Models through a Chemical Space Complementary DEL Screening Strategy; J. Med. Chem. 2024, 67, 18969-18980.

6. Qin S, Feng L, Zhao Q, Yan Z, Lyu X, Li K, Mu B, Chen Y, Lu W, Wang C, Suo Y, Yue J, Cui M, Li Y, Zhao Y*, Duan Z*, Zhu J*, Lu X*. Discovery and Optimization of WDR5 Inhibitors via Cascade Deoxyribonucleic Acid-Encoded Library Selection Approach. J Med Chem. 2024 67, 1079-1092.

7. Lulu Jiang, Sixiu Liu, Xinglong Jia, Qinting Gong, Xin Wen, Weiwei Lu, Jintong Yang, Xinyuan Wu, Xuan Wang, Yanrui Suo, Yilin Li, Motonari Uesugi, Zhi-bei Qu, Minjia Tan*, Xiaojie Lu* and Lu Zhou*，ABPP-CoDEL: Activity-Based Proteome Profiling-Guided Discovery of Tyrosine-Targeting Covalent Inhibitors from DNA-Encoded Libraries，J. Am. Chem. Soc. 2023, 46, 25283–25292

8. Wen X, Zhang M, Duan Z, Suo Y, Lu W, Jin R, Mu B, Li K, Zhang X, Meng L, Hong Y, Wang X, Hu H, Zhu J, Song W, Shen A*, Lu X*. Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)-one Focused DNA-Encoded Library. J Med Chem. 2023，66, 11118–11132 

9. Yang P, Wang X, Li B, Yang Y, Yue J, Suo Y, Tong H, He G, Lu X*, Chen G*. Streamlined construction of peptide macrocycles via palladium-catalyzed intramolecular S-arylation in solution and on DNA. Chem Sci. 2021, 12, 5804-5810.

10. Wang X, Liu J, Yan Z, Liu X, Liu S, Suo Y, Lu W, Yue J, Chen K, Jiang H, Zhao Y*, Zheng M*, Dai D*, Lu X*. Diversified strategy for the synthesis of DNA-encoded oxindole libraries. Chem Sci. 2021, 12, 2841-2847.